PI3K
PI3K (phosphatidylinositol-4,5-bisphosphate 3-kinase) is a family of enzymes involved in cellular functions such as cell growth, proliferation, differentiation, motility, survival and intracellular trafficking, which in turn are involved in cancer.
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A3268 CAL-130 HydrochlorideSummary: PI3K inhibitor
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A3340 CZC24832Summary: Selective PI3K-γ inhibitor
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A3432 GDC-0941 dimethanesulfonateSummary: PI3K inhibitor
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A3674 NVP-BKM120 HydrochlorideSummary: PI3K inhibitor
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A3724 PI-103 HydrochlorideTarget: PI3K|mTOR|DNA-PKSummary: DNA-PK/PI 3-kinase/mTOR inhibitor
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A3927 VS-5584 (SB2343)Target: PI3K|mTORSummary: MTOR/P13K inhibitor,potent and selective
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A4097 CUDC-907Target: Histone Deacetylases (HDACs)|PI3KSummary: Potent PI3K/HDAC inhibitor
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A3238 BEZ235 Tosylate1 CitationSummary: MTOR/P13K inhibitor
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B1047 GDC-0032Target: PI3KSummary: PI3Kα inhibitor
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B2186 GSK2636771Target: PI3KSummary: PIK3 inhibitor