EGFR
EGFR (epidermal growth factor receptor) is the cell-surface receptor of its specific ligands, including epidermal growth factor and TGFα (transforming growth factor α) and is a receptor tyrosine kinase.
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A8218 Lapatinib2 CitationTarget: ErbBSummary: EGFR/HER2 inhibitor,potent,selective and reversible
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A8319 Dacomitinib (PF299804, PF299)Target: ErbBSummary: HER inhibitor
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A8375 AZD8931 (Sapitinib)Target: EGFR|ErbBSummary: ErbB inhibitor
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A4092 CUDC-1011 CitationTarget: Histone Deacetylases (HDACs)|EGFR|ErbBSummary: Multitargeted HDAC inhibitor