Search results for: 'research area metabolism cyp3a cyp450'
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A3542 LCQ-908Summary: DGAT1 inhibitor
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A8202 Abiraterone acetateTarget: Cytochrome P450 (CYP450)Summary: Cytochrome p450 17a1 inhibitor
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A4240 Abiraterone1 CitationSummary: Potent CYP17 inhibitor
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A4302 Rosiglitazone maleateTarget: Insulin and Insulin-like ReceptorsSummary: PPARγ agonist,high-affinity and selective,potent insulin sensitizer
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A4303 GSK3787Summary: PPARβ/δ antagonist,novel and irreversible
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A4304 RosiglitazoneSummary: Potent PPARγ agonist
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A4307 GW0742Summary: PPARδ/β agonist,potent and selective
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A4311 PF-4981517Summary: CYP3A4 inhibitor,potent and selective
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A4316 KetoconazoleTarget: Cytochrome P450 (CYP450)Summary: Inhibitor of cyclosporine oxidase and testosterone 6 beta-hydroxylase
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A4317 Apremilast (CC-10004)Target: Phosphodiesterases (PDEs)Summary: PDE4 inhibitor