Androgen Receptor
AR (androgen receptor) is a member of steroid hormone receptor and ligand-activated transcription factor. It plays a crucial role in prostate cellular proliferation and male sexual differentiation.
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A8623 TOK-001Target: Androgen Receptors|Cytochrome P450 (CYP450)Summary: CYP17 inhibitor and androgen receptor (AR) antagonist
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A3003 MDV3100 (Enzalutamide)12 CitationTarget: Androgen ReceptorsSummary: Androgen receptor antagonist
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A5065 Bicalutamide1 CitationTarget: Androgen ReceptorsSummary: Androgen receptor antagonist
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A2150 AndarineTarget: Androgen ReceptorsSummary: Androgen receptor agonist
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A1372 AZD3514Summary: Androgen receptor downregulator
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B6041 EPI-001Summary: AR antagonist
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C3186 RD162Summary: androgen receptor (AR) antagonist
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C3546 HE-3235Summary: androgen receptor antagonist
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A8452 ODM-201Target: Androgen ReceptorsSummary: new-generation androgen receptor inhibitor
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C3644 DanazolSummary: weak androgenic effects