PI3K
PI3K (phosphatidylinositol-4,5-bisphosphate 3-kinase) is a family of enzymes involved in cellular functions such as cell growth, proliferation, differentiation, motility, survival and intracellular trafficking, which in turn are involved in cancer.
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A3724 PI-103 HydrochlorideTarget: PI3K|mTOR|DNA-PKSummary: DNA-PK/PI 3-kinase/mTOR inhibitor
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B1047 GDC-0032Target: PI3KSummary: PI3Kα inhibitor
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B2180 AS-252424Target: Akt|PI3KSummary: PI3Kγ inhibitor,novel and potent
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B2177 TG100713Target: PI3KSummary: pan-PI3K inhibitor
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A8488 NVP-BGT226Target: PI3K|mTORSummary: PI3K/mTOR inhibitor,selective and novel
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A8499 PF-04691502Target: Akt|PI3K|mTORSummary: PI3K/mTOR (FRAP) inhibitor
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A3005 CAL-101 (Idelalisib, GS-1101)2 CitationTarget: PI3KSummary: PI3K inhibitor
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A3015 BKM1201 CitationTarget: PI3KSummary: Inhibitor of pan-Class I PI3K
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B2176 GSK1059615Target: PI3K|mTORSummary: PI3K and mTOR inhibitor,potent and reversible
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A8210 GDC-094110 CitationTarget: PI3KSummary: PI3K inhibitor,potent and selective