Signaling Pathways
-
B3224 AZD3839Target: BACESummary: BACE1 inhibitor,potent and selective
-
B3225 BAF312 (Siponimod)1 CitationTarget: S1P receptorsSummary: S1P agonist,potent and selective
-
B3232 Z-IETD-FMK12 CitationTarget: CaspasesSummary: Caspase-8 inhibitor
-
B3233 Z-LEHD-FMK8 CitationTarget: CaspasesSummary: Irreversible Caspase-9 inhibitor.
-
B1372 Dorsomorphin 2HClSummary: AMPK inhibitor
-
B1383 VE-8222 CitationTarget: ATM/ATRSummary: ATR inhibitor
-
B1402 GZD824Target: Bcr-AblSummary: Bcr-Abl inhibitor,novel orally bioavailable
-
B1492 PYR-412 CitationTarget: ProteasomeSummary: inhibitor of Ubiquitin-Activating Enzyme (E1)
-
B1499 RVX-2082 CitationSummary: Potent BET bromodomain inhibitor
-
B1582 MM-1021 CitationSummary: MLL1 inhibitor,high-affinity peptidomimetic